| Identification | Back Directory | [Name]
(+)-JQ1 PA | [CAS]
2115701-93-2 | [Synonyms]
(+)-JQ1 PA
PubChem ID: 134821687
JQ1 PA;JQ-1 PA;JQ 1 PA
(6S)-4-(4-Chlorophenyl)-2,3,9-trimethyl-N-2-propyn-1-yl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine-6-acetamide
6H-Thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine-6-acetamide, 4-(4-chlorophenyl)-2,3,9-trimethyl-N-2-propyn-1-yl-, (6S)- | [Molecular Formula]
C22H20ClN5OS | [MDL Number]
MFCD31715451 | [MOL File]
2115701-93-2.mol | [Molecular Weight]
437.95 |
| Chemical Properties | Back Directory | [storage temp. ]
Store at -20°C | [solubility ]
DMF: 30 mg/ml; DMSO: 30 mg/ml; DMSO:PBS (pH 7.2) (1:6): 0.14 mg/ml; Ethanol: 25 mg/ml | [form ]
A crystalline solid |
| Hazard Information | Back Directory | [Biological Activity]
(+)-JQ1 PA is a derivative of the bromodomain and extra terminal domain (BET) inhibitor JQ1 with an IC50 value of 10.4 nM. | [in vitro]
(+)-JQ1 PA is a derivative of JQ1, which is the inhibitor of BET. The IC 50 of (+)-JQ1 PA for BET is 10.4 nM, and the IC 50 of JQ1 is 14.3 nM in MV4;11 cells. | [target]
| [storage]
Store at -20°C |
|
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