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BZ-VAL-GLY-ARG-AMC TRIFLUOROACETATE SALT

CAS No.
87779-49-5
Chemical Name:
BZ-VAL-GLY-ARG-AMC TRIFLUOROACETATE SALT
Synonyms
Bz-VGR-AMC;Bz-Val-Gly-Arg-AMC;BZ-VAL-GLY-ARG-AMC TFA SALT;Bz-Val-Gly-Arg-AMC (I-1085.0050);BZ-VAL-GLY-ARG-AMC TRIFLUOROACETATE SALT;N-Benzoyl-L-valylglycyl-N-(4-methyl-2-oxo-2H-1-benzopyran-7-yl)-L-argininamide;L-Argininamide, N-benzoyl-L-valylglycyl-N-(4-methyl-2-oxo-2H-1-benzopyran-7-yl)-;N-[(2S)-1-[[2-[[(2S)-5-(diaminomethylideneamino)-1-[(4-methyl-2-oxochromen-7-yl)amino]-1-oxopentan-2-yl]amino]-2-oxoethyl]amino]-3-methyl-1-oxobutan-2-yl]benzamide
CBNumber:
CB3241806
Molecular Formula:
C30H37N7O6
Molecular Weight:
591.66
MDL Number:
MFCD02259608
MOL File:
87779-49-5.mol
Last updated:2023-04-23 13:52:06

BZ-VAL-GLY-ARG-AMC TRIFLUOROACETATE SALT Properties

storage temp. -15°C
solubility Soluble in DMSO.
form White powder.
color White
Stability Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20° for up to 1 month.

BZ-VAL-GLY-ARG-AMC TRIFLUOROACETATE SALT price

Manufacturer Product number Product description CAS number Packaging Price Updated Buy
Biosynth Carbosynth FB110482 Bz-Val-Gly-Arg-AMC trifluoroacetate salt 87779-49-5 1mg $80 2021-12-16 Buy
Chem-Impex 32842 Bz-Val-Gly-Arg-AMC trifluoroacetate salt 87779-49-5 5MG $100 2021-12-16 Buy
Biosynth Carbosynth FB110482 Bz-Val-Gly-Arg-AMC trifluoroacetate salt 87779-49-5 2mg $125 2021-12-16 Buy
Biosynth Carbosynth FB110482 Bz-Val-Gly-Arg-AMC trifluoroacetate salt 87779-49-5 5mg $200 2021-12-16 Buy
Biosynth Carbosynth FB110482 Bz-Val-Gly-Arg-AMC trifluoroacetate salt 87779-49-5 10mg $320 2021-12-16 Buy
Product number Packaging Price Buy
FB110482 1mg $80 Buy
32842 5MG $100 Buy
FB110482 2mg $125 Buy
FB110482 5mg $200 Buy
FB110482 10mg $320 Buy

BZ-VAL-GLY-ARG-AMC TRIFLUOROACETATE SALT Chemical Properties,Uses,Production

Description

Bz-VGR-AMC (87779-49-5) may be used for measuring the trypsin-like activity of the 20S proteasome, in combination with Suc-LLVY-AMC (Cat.# 10-2971, for assaying its chymotrypsin-like activity) and Z-LLE-AMC, (for determining its PGPH activity). Fluorogenic substrate. Ex.: 380nm Em.: 460nm.

Uses

Bz-Val-Gly-Arg-AMC is a bioactive compound used in assaying the degree of inhibition conferred by PS-341, a potent peptidylboronic acid with anticancer properties.

References

1) Gillardon?et al. (2007),?The 20S proteasome isolated from Alzheimer’s disease brain shows post-translational modifications but unchanged proteolytic activity; J. Neurochem.,?101?1483 2) Kim?et al. (2002),?Navigation inside a protease: substrate selection and product exit in tricorn protease from Thermoplasma acidophilum; J. Mol. Biol.,?324?1041 3) Dahlmann?et al. (2000),?Different proteasome subtypes in a single tissue exhibit different enzymatic properties; J. Mol. Biol.,?303?643 4) Lightcap?et al. (2000),?Proteasome inhibition measurements: clinical application; Clin. Chem.,?46?673

BZ-VAL-GLY-ARG-AMC TRIFLUOROACETATE SALT Preparation Products And Raw materials

Raw materials

Preparation Products

BZ-VAL-GLY-ARG-AMC TRIFLUOROACETATE SALT Suppliers

Global( 44)Suppliers
Supplier Tel Email Country ProdList Advantage
Chengdu Youngshe Chemical Co., Ltd.
+8618108235634 Cecilia@youngshechem.com China 2345 58
LEAP CHEM CO., LTD.
+86-852-30606658 market18@leapchem.com China 24738 58
Nanjing TGpeptide
+86-13347807150 +86-13347807150 support@tgpeptide.com China 3279 58
Aladdin Scientific
+1-833-552-7181 sales@aladdinsci.com United States 52927 58
GL Biochem (Shanghai) Ltd 21-61263452 13641803416 ymbetter@glbiochem.com China 9981 64
Shanghai Hanhong Scientific Co.,Ltd. 021-021-64543801 13764082696 2355241799@qq.com China 42982 64
Chemsky (shanghai) International Co.,Ltd 021-50135380 shchemsky@sina.com China 15421 60
Nanjing Leon Biological Technology Co., Ltd. 17705183659 sales@njleonbiotech.com China 5503 55
Nanjing Peptide Biotech Ltd. 025-025-58361106-805-805 13082558573 liugang@njpeptide.com China 9962 55
Hangzhou Peptidego Biotech Co.,Ltd. 0571-87213919 eric@peptidego.com China 6347 58
BZ-VAL-GLY-ARG-AMC TFA SALT BZ-VAL-GLY-ARG-AMC TRIFLUOROACETATE SALT Bz-VGR-AMC Bz-Val-Gly-Arg-AMC N-[(2S)-1-[[2-[[(2S)-5-(diaminomethylideneamino)-1-[(4-methyl-2-oxochromen-7-yl)amino]-1-oxopentan-2-yl]amino]-2-oxoethyl]amino]-3-methyl-1-oxobutan-2-yl]benzamide L-Argininamide, N-benzoyl-L-valylglycyl-N-(4-methyl-2-oxo-2H-1-benzopyran-7-yl)- N-Benzoyl-L-valylglycyl-N-(4-methyl-2-oxo-2H-1-benzopyran-7-yl)-L-argininamide Bz-Val-Gly-Arg-AMC (I-1085.0050) 87779-49-5 C30H37N7O6 Miscellaneous Enzyme